Organic compounds -- part of the class 532-570 series inventions 03/09

20090082568 - Accelerated reduction of organic substances with boranes: In a process for the accelerated reduction of organic substrates, selected from the group consisting of ester, amides, nitriles, acids, ketones, imines or mixtures thereof, the substrates are reacted with an amine borane, sulfide borane or ether borane complex as a borane source in the presence of organic accelerator compounds... Agent: Connolly Bove Lodge & Hutz, LLP

20090082569 - Narcistatin prodrugs: The present invention provides prodrugs derived from the sparingly soluble anticancer isocarbostyril narciclasine, a component of various Narcissus species, said prodrugs having potential for use against animal and human cancers. Also disclosed is an efficient procedure for the synthetic conversion of narciclasine to several more soluble cyclic phosphate compounds, including... Agent: Fennemore Craig

20090082570 - Method of manufacturing bipyridinium compound and synthetic intermediate of the same, method of manufacturing dye compound, and novel bipyridinium compound and novel dye compound comprising the same: In general formula (A), Ar1 and Ar2 each independently denote an optionally substituted (hetero)aryl group, R3 and R4 each independently denote a substituent that may form a ring with a pyridine ring to which the substituent substitutes, m3 and m4 each independently denote an integer ranging from 0 to 4,... Agent: Sughrue Mion, PLLC

20090082571 - Intermediates of 2-substituted carbapenem derivatives and process for production thereof: The present invention relates to compounds represented by formula (1) and a process for producing the same. The use of these compounds can realize the production of carbapenem derivatives having potent antimicrobial activity and a wide antimicrobial spectrum in a safe and cost-effective manner.... Agent: Wenderoth, Lind & Ponack, L.L.P.

20090082572 - Process for amorphous esomeprazole: The present invention relates to a commercially viable process for preparation of amorphous esomeprazole. Thus, amorphous esomeprazole is prepared by suspending esomeprazole in water and then subjecting the suspension to lyophilization at −70° C.... Agent: Caesar, Rivise, Bernstein, Cohen & Pokotilow, Ltd.

20090082573 - Methods for preparation of pyridylamines: Alternate methods for preparing functionalized pyridyl-amine products from pyridinyl starting materials are provided herein. In addition, these alternately-prepared functionalized pyridyl-amines can be used as ligands or ligand precursors in catalytic compositions, e.g. for use in alkene oligomerization reactions.... Agent: Exxonmobil Chemical Company

20090076275 - Diacylglycerol acyltransferase inhibitors: P

20090076276 - Isoquinoline compound and pharmaceutical use thereof:

20090076277 - Process for the preparation of pyridine-methylsulfinyl compounds: wherein Q, R1-R7 are as herein defined; with a reducing agent selected from a trivalent phosphorous compound, an oxidizable solvent and a sulfonic acid chloride; and, if desired, the conversion of a compound of formula (I) to another compound of formula (I) or a salt thereof.... Agent: Griffin & Szipl, PC

20090069564 - Methods and compositions for selectin inhibition: P

20090069565 - New indole derivatives as factor xa inhibitors: in which R0; R1; R2; R3; R4; R5; R6; R7; Q; V, G and M have the meanings indicated in the claims. The compounds of formula I are valuable pharmacologically active compounds. They exhibit a strong antithrombotic effect and are suitable, for example, for the therapy and prophylaxis of cardiovascular... Agent: Andrea Q. Ryan Sanofi-aventis U.s. LLC

20090062542 - Novel red electroluminescent compounds and organic electroluminescent device using the same: The present invention relates to novel red phosphorescent compounds exhibiting high luminous efficiency, and organic electroluminescent devices comprising the same.... Agent: Edwin Oh Rohm And Haas Electronic Materials LLC

20090062543 - Uv excitable fluorescent energy transfer dyes: Novel energy transfer dyes which can be used with shorter wavelength light sources are provided. These dyes include a donor dye with an absorption maxima at a wavelength between about 250 to 450 nm and an acceptor dye which is capable of absorbing energy emitted from the donor dye. One... Agent: Dechert LLP

20090062544 - Crystals of morphinan derivative and process for producing the same: The present invention is directed to provide 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-[N-methyl-trans-3-(3-furyl)acrylamido]morphinan hydrochloride consistent in quality after production and having high purity. A crystal of 17-cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-[N-methyl-trans-3-(3-furyl)acrylamido]morphinan hydrochloride including a A-form, B-form or C-form crystal thereof, and a process for producing the same are provided.... Agent: Birch Stewart Kolasch & Birch

20090062545 - Trisazo compound, ink composition, recording method, and colored article: R2 represents a cyano group, a carbamoyl group or a carboxy group, each of R3 and R4 independently represents a hydrogen atom, a methyl group, a chlorine atom or a sulfo group, respectively) and a water-based black ink composition containing said compound; said compound has high solubility in a medium... Agent: Nields & Lemack

20090062546 - Dolasetron trifluoroacetate, polymorphs of dolasetron trifluoroacetate and process for preparation thereof: Provided are crystalline forms of dolasetron trifluoroacetate, methods for their preparation, and their use in preparing dolasetron mesylate.... Agent: Kenyon & Kenyon LLP

20090062547 - Cyclic-fused beta-lactones and their synthesis: The present invention provides a concise synthetic method for generating lactam-fused beta-lactones that feature, in some embodiments, a tertiary fused carbinol, quaternary carbons, and a reactive beta-lactone moiety available for further reactions. The present invention further provides compounds synthesized by this method as well as methods of using these compounds... Agent: Fulbright & Jaworski L.L.P.

20090062548 - Novel pyridine oxide compound, and process for producing carboxylic acid derivative and optically active carboxylic acid derivative with the use of the same: The invention relates to a pyridine oxide compound represented by formula (I), an optically active compound thereof, a salt thereof and a hydrate thereof, and, in the presence of the compound as a catalyst, performing 1) a method for producing an ester compound or an amide compound from a carboxylic... Agent: Thomas, Kayden, Horstemeyer & Risley, LLP